Chemistry and Structure of Mitomycin C Calvin L. Stevens, K. Grant Taylor, Morton E. Munk, W. S. Marshall, Klaus Noll, G. D. Shah, L. G. Shah, and K. Uzu pp 1 - 10; DOI: 10.1021/jm00325a001 |
Potential Anticancer Agents. II. The Synthesis of Some Nitrogen Mustard Containing Sulfones and Thiosulfinates Allen F. Hirsch, Claude Piantadosi, and J. Logan Irvin pp 10 - 14; DOI: 10.1021/jm00325a002 |
Enzyme-Alterable Alkylating Agents. VII. The Design of Short-Lived Mustards Samuel Sass, Charles E. Williamson, Stanley P. Kramer, Louis E. Goodman, Adolph Ulfohn, Arnold M. Seligman, and Benjamin Witten pp 14 - 17; DOI: 10.1021/jm00325a003 |
Structure Studies on Vancomycin Frederick J. Marshall pp 18 - 22; DOI: 10.1021/jm00325a004 |
The Chemistry of Cephalosporin Antibiotics. III. Acylation of Cephalosporadesates Earle Van Heyningen pp 22 - 25; DOI: 10.1021/jm00325a005 |
Syntheses with 5-Nitro-2-furonitrile W. R. Sherman and Anne Von Esch pp 25 - 28; DOI: 10.1021/jm00325a006 |
Potential Antiradiation Drugs. I. Amide, Hydroxamic Acid, and Hydrazine Derivatives of Mercapto Acids. Amino Thioacids Edward R. Atkinson, G. Richard Handrick, Robert J. Bruni, and Felix E. Granchelli pp 29 - 33; DOI: 10.1021/jm00325a007 |
Enzyme Inhibitors. VI. Studies on the Bulk Tolerance of Adenosine Deaminase for 6-Substituted Amino-9-(3-hydroxypropyl)purines Howard J. Schaeffer and Robert Vince pp 33 - 35; DOI: 10.1021/jm00325a008 |
Analogs of Tetrahydrofolic Acid. XVII.1,2 On the Mode of Binding of the p-Aminobenzoyl Moiety of N-(2-Amino-4-hydroxy-6-methyl-6-pyrimidylpropyl)-p-aminobenzoyl- L-glutamic Acid to Dihydrofolic Reductase B. R. Baker and Johannes H. Jordaan pp 35 - 41; DOI: 10.1021/jm00325a009 |
Synthesis of Fatty Acids with Smooth Muscle Stimulant Activity E. Crundwell, M. A. Pinnegar, and W. Templeton pp 41 - 45; DOI: 10.1021/jm00325a010 |
Hypocholesterolemic Agents. V.1a Isomeric Azacholesterols1b R. E. Counsell, P. D. Klimstra, L. N. Nysted, and R. E. Ranney pp 45 - 48; DOI: 10.1021/jm00325a011 |
Anabolic Agents. A-Ring Conjugated Enone Androstane Derivatives P. D. Klimstra and R. E. Counsell pp 48 - 52; DOI: 10.1021/jm00325a012 |
Mammalian Antifertility Agents. I. Derivatives of 2,3-Diphenylindenes Daniel Lednicer, John C. Babcock, Paul E. Marlatt, Stanley C. Lyster, and Gordon W. Duncan pp 52 - 57; DOI: 10.1021/jm00325a013 |
Studies in Alkyl-Oxygen Heterolysis. Some 4-Alkoxypiperidines Related to Reversed Esters of Pethidine A. F. Casy and N. A. Armstrong pp 57 - 61; DOI: 10.1021/jm00325a014 |
Spiranes. VII. Neuroleptics Derived from Azaspiranes Charles H. Grogan, Charles F. Geschickter, Meier E. Freed, and Leonard M. Rice pp 62 - 73; DOI: 10.1021/jm00325a015 |
Derivatives of Morphanthridine L. H. Werner, S. Ricca, E. Mohacsi, A. Rossi, and V. P. Arya pp 74 - 80; DOI: 10.1021/jm00325a016 |
The Synthesis and Pharmacology of Some Substituted 1,3-Benzodioxoles and 1,4-Benzodioxans M. W. Baines, D. B. Cobb, R. J. Eden, R. Fielden, J. N. Gardner, A. M. Roe, W. Tertiuk, and G. L. Willey pp 81 - 90; DOI: 10.1021/jm00325a017 |
Diuretics. 6-Substituted 3-Ketoalkyl-3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-Dioxides and Related Anils, Oximes, and Hydrazones Jerry E. Robertson, Donald A. Dusterhoft, and Thomas F. Mitchell pp 90 - 95; DOI: 10.1021/jm00325a018 |
Behavioral Stimulants. 4-Oxazolidinones John B. Bicking, Sara F. Kwong, Michael H. Fisher, and William H. Nicholson pp 95 - 100; DOI: 10.1021/jm00325a019 |
Behavioral and Neuropharmacological Actions of N-Aralkylhydroxylamines and Their O-Methyl Ethers F. Benington, R. D. Morin, and L. C. Clark pp 100 - 104; DOI: 10.1021/jm00325a020 |
Synthesis and Pharmacological Study of New Piperazine Derivatives. II. Phenethylpiperazines R. Ratouis, J. R. Boissier, and C. Dumont pp 104 - 107; DOI: 10.1021/jm00325a021 |
p-Amino-N-[2-(substituted amino)ethyl]benzamides. Potential Antifibrillatory Drugs Per Thyrum and Allan R. Day pp 107 - 111; DOI: 10.1021/jm00325a022 |
Pyridoxine Chemistry. VI. Homologs of Pyridoxol and of 5-Pyridoxic Acid W. Korytnyk pp 112 - 115; DOI: 10.1021/jm00325a023 |
Pyridoxine Chemistry. VII.1a Some Modifications in the 4-Position of Pyridoxol1b R. P. Singh and W. Korytnyk pp 116 - 117; DOI: 10.1021/jm00325a024 |
Substitution in the Hydantoin Ring. I. N-3-Aminomethyl Derivatives Meldrum B. Winstead, Donald E. Barr, Coleman R. Hamel, D. James Renn, Harriet I. Parker, and Richard M. Neumann pp 117 - 120; DOI: 10.1021/jm00325a025 |
Substitution in the Hydantoin Ring. II. N-3-Acetic Acid Derivatives Meldrum B. Winstead and Coleman R. Hamel pp 120 - 122; DOI: 10.1021/jm00325a026 |
N,N-Diethyl-2,2-dimethylpropane-1,3-diamine Morris Freifelder and Yew Hay Ng pp 122 - 123; DOI: 10.1021/jm00325a027 |
Derivatives of Morphine. IV.1 14-Hydroxymorphine and 14-Hydroxydihydromorphine Ulrich Weiss and Sol J. Daum pp 123 - 125; DOI: 10.1021/jm00325a028 |
1,2,3,4-Tetrahydroisoquinoline Derivatives with Antihypertensive Properties Wilhelm Wenner pp 125 - 126; DOI: 10.1021/jm00325a029 |
N-Ethoxy-4-ethylamino-3-methyl-2-phenyl-2-propionoxy-1-α-pyridylbutane. An Analog of the Analgesic Propoxyphene Randolph T. Major, Konrad Fitzi, and Hans-Jürgen Hess pp 127 - 129; DOI: 10.1021/jm00325a030 |
Synthesis and Pharmacological Study of Pyridazines. I. Alkoxypyridazines Peter Coad, Raylene Adams Coad, Barry Dubinsky, Joseph P. Buckley, and William Kinnard pp 129 - 131; DOI: 10.1021/jm00325a031 |
Novel Oral Hypoglycemic Agents. I. Hexahydroindeno[1,2-c]pyrroles and Indanamines Samir Chandra Lahiri and Balai Pathak pp 131 - 133; DOI: 10.1021/jm00325a032 |
17α-Methylandrostane-3α,17β-diol K. R. Bharucha and F. M. Martin pp 133 - 136; DOI: 10.1021/jm00325a033 |
Benzo[b]thiophene Derivatives. V. Mannich Bases With Antimicrobial Activity E. Campaigne, E. D. Weinberg, G. Carlson, and E. S. Neiss pp 136 - 137; DOI: 10.1021/jm00325a034 |
4-(Alkoxystyryl)quinolines C. T. Bahner, H. Kinder, and T. Rigdon pp 137 - 138; DOI: 10.1021/jm00325a035 |
The Purification of Aminopterin Ti Li Loo pp 139 - 139; DOI: 10.1021/jm00325a036 |
Some 3,4,5-Trimethoxy-Substituted Benzamides S. K. Sogani and P. C. Dandiya pp 139 - 140; DOI: 10.1021/jm00325a037 |
1-(2-Deoxy-D-glucopyranosyl)-5-fluorocytosine George J. Durr pp 140 - 141; DOI: 10.1021/jm00325a038 |
Some Bis(3-nitro- and 3-amino-4-alkoxy- and -4-aryloxyphenyl) Sulfones William F. Hart and Martin E. McGreal pp 141 - 142; DOI: 10.1021/jm00325a039 |
A Convenient Synthesis of Aminotryptamines Analogous to Serotonin S. P. Hiremath and S. Siddappa pp 142 - 143; DOI: 10.1021/jm00325a040 |
New Derivatives of 9-Amino-1,2,3,4-tetrahydroacridine W. P. Brian and B. L. Souther pp 143 - 144; DOI: 10.1021/jm00325a041 |
7- and 12-(o-Halophenyl)benz[a]anthracenes Frank A. Vingiello, Leo Ojakaar, and Rosalie Kelsey pp 144 - 144; DOI: 10.1021/jm00325a042 |
Survey of Chemical Notation Systems Frederick Y. Wiselogle pp 145 - 145; DOI: 10.1021/jm00325a043 |
Advances in Chemotherapy. Volume I. Alfred Burger pp 145 - 145; DOI: 10.1021/jm00325a044 |
The Background to Chemotherapy of Virus Diseases Alfred Burger pp 145 - 145; DOI: 10.1021/jm00325a045 |
Research Progress in Organic--Biological and Medicinal Chemistry. Volume I. Alfred Burger pp 146 - 146; DOI: 10.1021/jm00325a046 |
Progress in Drug Research. Volume 7. Alfred Burger pp 146 - 146; DOI: 10.1021/jm00325a047 |
Experimental Chemotherapy. Volume III. Chemotherapy of Bacterial Infections. Part II. Chemotherapy of Fungal, Rickettsial, and Viral Infections Alfred Burger pp 146 - 146; DOI: 10.1021/jm00325a048 |
Stereochemical Studies on Medicinal Agents. II. Absolute Configuration of (-)-Phenampromide Philip S. Portoghese pp 147 - 150; DOI: 10.1021/jm00326a001 |
Substituent Constants for Aliphatic Functions Obtained from Partition Coefficients Junkichi Iwasa, Toshio Fujita, and Corwin Hansch pp 150 - 153; DOI: 10.1021/jm00326a002 |
The Formation of O-Methylated Catechols by Microsomal Hydroxylation of Phenols and Subsequent Enzymatic Catechol O-Methylation. John Daly, Joseph K. Inscoe, and Julius Axelrod pp 153 - 157; DOI: 10.1021/jm00326a003 |
Excretion, Distribution, and Metabolism of Doxapram Hydrochloride Robert B. Bruce, J. E. Pitts, Franklin Pinchbeck, and Jack Newman pp 157 - 164; DOI: 10.1021/jm00326a004 |
A Simple Test Tube Arrangement for Screening Fibrinolytic Activity of Synthetic Organic Compounds Kurt N. von Kaulla pp 164 - 166; DOI: 10.1021/jm00326a005 |
A Study of Comparative Chemical and Biological Activities of Alkylating Agents T. J. Bardos, N. Datta-Gupta, P. Hebborn, and D. J. Triggle pp 167 - 174; DOI: 10.1021/jm00326a006 |
The Chemistry of Cephalosporins. IV. Acetoxyl Replacements with Xanthates and Dithiocarbamates Earle Van Heyningen and Carter N. Brown pp 174 - 181; DOI: 10.1021/jm00326a007 |
Synthesis and Antitumor Activity of 9-Substituted Nitrogen Mustard Derivatives of 6-Alkylthiopurines Darrell E. O'Brien, James D. Westover, Roland K. Robins, and C. C. Cheng pp 182 - 187; DOI: 10.1021/jm00326a008 |
Nitrogen Mustards Derived from 3,4-Dihydro-2,4-dioxo-1(2H)-pyrimidinepropionic and -butyric Acids Abelardo P. Martinez, William W. Lee, and Leon Goodman pp 187 - 189; DOI: 10.1021/jm00326a009 |
Purine N-Oxides. XV. The Synthesis of 6-Mercaptopurine 3-N-Oxide. Its Chemotherapeutic Possibilities George Bosworth Brown, Gershon Levin, Sarah Murphy, Alex Sele, H. Christine Reilly, George S. Tarnowski, Franz A. Schmid, Morris N. Teller, and C. Chester Stock pp 190 - 195; DOI: 10.1021/jm00326a010 |
Pyrimidinecarbamates and Thiolcarbamates Derived from Amino- and Oxopyrimidines. II Elizabeth Dyer and Henry Richmond pp 195 - 200; DOI: 10.1021/jm00326a011 |
Acyltryptamines. IV.1 Azepino[5,4,3-cd]indoles Maximilian von Strandtmann, Marvin P. Cohen, and John Shavel pp 200 - 204; DOI: 10.1021/jm00326a012 |
1-p-Chlorobenzyl-5-methylindole-3-acetic Acid. Some 2-Substituted Derivatives Edward Walton, Charles H. Stammer, Ruth F. Nutt, Susan R. Jenkins, and Frederick W. Holly pp 204 - 208; DOI: 10.1021/jm00326a013 |
Thio Analogs of Carisoprodol (N-Isopropyl-2-methyl-2-propyl-1,3-propanediol Dicarbamate) M. A. Leaffer, W. A. Skinner, and B. J. Ludwig pp 208 - 212; DOI: 10.1021/jm00326a014 |
Adrenal Cortical Inhibitors and Potent Synthetic Estrogens W. L. Bencze, L. I. Barsky, W. P. Sopchak, A. A. Renzi, N. Howie, and J. J. Chart pp 213 - 214; DOI: 10.1021/jm00326a015 |
The Modification of 11β-Hydroxy-11α-methyl-5β-pregnane-3,20-dione Dioxime under Acidic Conditions Donald R. Buhler, Louis C. Schroeter, and W. J. Wechter pp 215 - 219; DOI: 10.1021/jm00326a016 |
DL-1-(1-Arylalkyl)imidazole-5-carboxylate Esters. A Novel Type of Hypnotic Agents Erik F. Godefroi, Paul A. J. Janssen, Cyriel A. M. Van der Eycken, Albert H. M. T. Van Heertum, and Carlos J. E. Niemegeers pp 220 - 223; DOI: 10.1021/jm00326a017 |
Hypocholesteremic Agents. III.1 Basic Carbinols and Related Compounds James H. Short, Ursula Biermacher, Daniel A. Dunnigan, G. Frederick Lambert, Donald L. Martin, Carl W. Nordeen, and Howard B. Wright pp 223 - 230; DOI: 10.1021/jm00326a018 |
The Synthesis of Phencyclidine and Other 1-Arylcyclohexylamines V Harold Maddox, Erik F. Godefroi, and Robert F. Parcell pp 230 - 235; DOI: 10.1021/jm00326a019 |
Structures Related to Morphine. XXVIII.1 Alternative Syntheses of α- and β-2,9-Dimethyl-2′-hydroxy-5-propyl-6,7-benzomorphan Colin F. Chignell, J. Harrison Ager, and Everette L. May pp 235 - 238; DOI: 10.1021/jm00326a020 |
The Chemistry and Pharmacology of a Series of Cycloalkanespiro-5′-hydantoins W. Oldfield and C. H. Cashin pp 239 - 249; DOI: 10.1021/jm00326a021 |
Synthetic Antigonadotropins. III H. H. Fox, J. T. Gibas, H. L. Lee, and A. Boris pp 250 - 251; DOI: 10.1021/jm00326a022 |
Synthesis of 6- and 7-Bis(2-chloroethyl)amino-DL-tryptophan Leon Goodman, Roland R. Spencer, Giovanni Casini, Osborne P. Crews, and Elmer J. Reist pp 251 - 252; DOI: 10.1021/jm00326a023 |
Carcinogenic Activity of 2-N,N-Dimethylamino-5-phenylazopyridine Ellis V. Brown, Andrew F. Smetana, and Ali A. Hamdan pp 252 - 253; DOI: 10.1021/jm00326a024 |
Some 5-Fluoropyrimidines G. J. Durr pp 253 - 255; DOI: 10.1021/jm00326a025 |
New 1-Aminomethylbenzocyclobutenes Joseph A. Skorcz and Jerry E. Robertson pp 255 - 257; DOI: 10.1021/jm00326a026 |
A New Group of Antifibrillants. N-(ω-Aminoalkyl)phthalimides Kálmán Hideg and H. Olga Hankovszky pp 257 - 259; DOI: 10.1021/jm00326a027 |
The Synthesis of Ethyl α-(p-Chlorophenyl)-6,7-dimethoxy-2-methyl- 1,2,3,4-tetrahydro-1-isoquinolinepropionate Glenn C. Morrison and John Shavel pp 259 - 260; DOI: 10.1021/jm00326a028 |
Synthesis and Biological Activities of Certain Short-Chain Mono- and Bisquaternary Ammonium Compounds Walter L. Graef, Joseph G. Cannon, and Joseph P. Buckley pp 260 - 263; DOI: 10.1021/jm00326a029 |
1,3,2-Diazaphosphorinane 2-Oxides. II.1 Synthesis of Some 1,3-Bis(aralkyl)-2-(N-arylamino)-1,3,2-diazaphosphorinane 2-Oxides2 John H. Billman and John L. Meisenheimer pp 264 - 265; DOI: 10.1021/jm00326a030 |
Hexahydro-11H-pyrrolo[2,1-α]-β-carbolines and Tetrahydro-13H-isoindolo[1,2-α]-β-carbolines S. Wawzonek and J. D. Nordstrom pp 265 - 267; DOI: 10.1021/jm00326a031 |
A Carbocyclic Analog of Glyceraldehyde Dimer James G. Murphy pp 267 - 268; DOI: 10.1021/jm00326a032 |
The Preparation and Some Biological Properties of 17α-Ethyl-17β-methyl-Δ4,13-gonadien-3-one R. Y. Kirdani and R. I. Dorfman pp 268 - 269; DOI: 10.1021/jm00326a033 |
Hydroxy-, Nitro-, Amino-, and Methoxy-4-(4-dimethylaminostyryl)quinolines Carl Tabb Bahner, David Brotherton, William H. Chapman, William Longmire, H. Bernie Orr, Lydia Moore Rives, Emma Brown Senter, and Warren Yee pp 269 - 271; DOI: 10.1021/jm00326a034 |
Synthesis and Pharmacological Study of New Piperazine Derivatives. III. Phenoxyalkylpiperazines R. Ratouis, J. R. Boissier, and C. Dumont pp 271 - 273; DOI: 10.1021/jm00326a035 |
Synthesis of Tripeptides of 1-Aminocyclopentane-1-carboxylic Acid J. Friedrich Diehl and David O. Bowen pp 274 - 274; DOI: 10.1021/jm00326a036 |
An Improved Synthesis of Oxotremorine Alan Bebbington and Derek Shakeshaft pp 274 - 275; DOI: 10.1021/jm00326a037 |
Perchloric Acid in the Preparation of 2′,3′-Isopropylidene 6-Thioinosine John A. Zderic, John G. Moffatt, Don Kau, Koert Gerzon, and William E. Fitzgibbon pp 275 - 275; DOI: 10.1021/jm00326a038 |
Synthesis of Some Amino Acid Thiol Esters Robert A. Ray and Robert B. Johnston pp 275 - 276; DOI: 10.1021/jm00326a039 |
Advances in Drug Research. Volume 1. Alfred Burger pp 277 - 277; DOI: 10.1021/jm00326a040 |
Molecular Modification in Drug Design. Alfred Burger pp 277 - 277; DOI: 10.1021/jm00326a041 |
Science Citation Index. Volume 1, 1964. Wilhelm Moll pp 277 - 278; DOI: 10.1021/jm00326a042 |
Pharmaceutical Microbiology. Charles J. Paget pp 278 - 278; DOI: 10.1021/jm00326a043 |
Handbook of Chemistry and Physics. Alfred Burger pp 278 - 278; DOI: 10.1021/jm00326a044 |
CORRECTION pp 278 - 278; DOI: 10.1021/jm00326a045 |
Structure-Activity Relationships in the Field of Antibacterial Steroid Acids Josef Fried, Gerald W. Krakower, David Rosenthal, and Harold Basch pp 279 - 282; DOI: 10.1021/jm00327a001 |
Analogs of Tetrahydrofolic Acid. XVIII.1,2 On the Mode of Binding of Some 6-Aryl- and 6-Aralkylpyrimidines to Folic Reductase B. R. Baker, Howard S. Shapiro, and William C. Werkheiser pp 283 - 287; DOI: 10.1021/jm00327a002 |
Amino Acid Analogs of Tryptamine Antagonists of Serotonin Frederick Leonard and Walter Tschannen pp 287 - 290; DOI: 10.1021/jm00327a003 |
2-Amino-3-methylthiobutyric Acid, an Isoleucine Antagonist Tommy J. McCord, Drusilla Cook Howell, Don L. Tharp, and Alvie L. Davis pp 290 - 292; DOI: 10.1021/jm00327a004 |
Synthesis of Some Pyrimidine Amino Acids by the Rhodanine Method and Tests vs. the Ehrlich Ascites Carcinoma Vilhjalmur G. Skulason, Claude Piantadosi, Benjamin F. Zamberana, and J. Logan Irvin pp 292 - 295; DOI: 10.1021/jm00327a005 |
Synthesis and Structure-Activity Relationships of Some Aminopyridines, Imidazopyridines, and Triazolopyridines M. M. Vohra, S. N. Pradhan, P. C. Jain, S. K. Chatterjee, and Nitya Anand pp 296 - 304; DOI: 10.1021/jm00327a006 |
Derivatives of Imidazole. I. Synthesis and Reactions of Imidazo[1,2-α]pyridines with Analgesic, Antiinflammatory, Antipyretic, and Anticonvulsant Activity Luigi Almirante, Luigi Polo, Alfonso Mugnaini, Ercolina Provinciali, Pierluigi Rugarli, Adriana Biancotti, Afro Gamba, and Walter Murmann pp 305 - 312; DOI: 10.1021/jm00327a007 |
3-Alkyl-3-phenylpiperidine Derivatives as Analgesics. II Hiroshi Kugita, Toyonari Oine, Hirozumi Inoue, and Goro Hayashi pp 313 - 316; DOI: 10.1021/jm00327a008 |
Analgetics Based on the Pyrrolidine Ring. IV J. F. Cavalla, D. C. Bishop, R. A. Selway, N. E. Webb, C. V. Winder, and M. Welford pp 316 - 326; DOI: 10.1021/jm00327a009 |
Bicyclic Homologs of Piperazine. VII.1 Synthesis and Analgesic Activity of 3-Aralkenyl-8-propionyl-3,8-diazabicyclo[3.2.1]octanes Giorgio Cignarella, Emilio Occelli, and Emilio Testa pp 326 - 331; DOI: 10.1021/jm00327a010 |
N,N′-Disubstituted Compounds with Diverse Biological Activities Robert P. Mull, Carl Tannenbaum, Mary R. Dapero, Marcel Bernier, William Yost, and George DeStevens pp 332 - 338; DOI: 10.1021/jm00327a011 |
Yohimbane Derivatives. II. The Synthesis and Psychopharmacological Properties of Yohimbane Derivatives with Halogen Substitutents in Ring E Maximilian von Strandtmann, George Bobowski, and John Shavel pp 338 - 341; DOI: 10.1021/jm00327a012 |
Triptycene Derivatives as Medicinal Agents Edmund C. Kornfeld, Pam Barney, John Blankley, and William Faul pp 342 - 347; DOI: 10.1021/jm00327a013 |
Derivatives of Fluorene. XIX.1,2 9-o-Chlorocinnamylidenefluorene and Related Compounds T. Lloyd Fletcher, Moses J. Namkung, John R. Dice, and Sandra K. Schaefer pp 347 - 350; DOI: 10.1021/jm00327a014 |
5-Methylpyrazole-3-carboxylic Acid. The Potent Hypoglycemic Metabolite of 3,5-Dimethylpyrazole in the Rat David L. Smith, Arlington A. Forist, and William E. Dulin pp 350 - 353; DOI: 10.1021/jm00327a015 |
The Effects of Ring-Methoxyl Groups on Biological Deamination of Phenethylamines Leland C. Clark, Frederick Benington, and Richard D. Morin pp 353 - 355; DOI: 10.1021/jm00327a016 |
Some Cardiovascular Effects of a Series of Aryloxyalkylamines. I J. Augstein, W. C. Austin, R. J. Boscott, S. M. Green, and C. R. Worthing pp 356 - 367; DOI: 10.1021/jm00327a017 |
Ultraviolet Absorption Spectra and Apparent Acidic Dissociation Constants of Some Phenolic Amines Thomas Kappe and Marvin D. Armstrong pp 368 - 374; DOI: 10.1021/jm00327a018 |
Antifungal Activity of a Series of Substituted [(α-Nitroalkyl)benzylthio]alkylamines Robert C. Tweit, R. D. Muir, Seth Mizuba, and Webster R. Crowley pp 374 - 377; DOI: 10.1021/jm00327a019 |
Phosphorylated Benzenesulfonamides as Animal Systemic Insecticides Frank A. Wagner, Ronald W. Baer, and Gerald Berkelhammer pp 377 - 383; DOI: 10.1021/jm00327a020 |
Spiro-3-oxiranyl-5α-androstan-17β-ols H. G. Lehmann, O. Engelfried, and R. Wiechert pp 383 - 384; DOI: 10.1021/jm00327a021 |
Structures Related to Morphine. XXIX.1 Further Experiments on the Stereo-Controlled Reduction of 9-Methylene-6,7-benzomorphans Colin F. Chignell and Everette L. May pp 385 - 386; DOI: 10.1021/jm00327a022 |
Synthesis of 17-Acetoxy-6-chloro-21-fluoropregna-4,6-diene-3,20-dione, a Highly Active Oral Progestin Robert F. R. Church and Martin J. Weiss pp 386 - 387; DOI: 10.1021/jm00327a023 |
2H-1,3,2-Oxazaphosphorine Derivatives Carl Tabb Bahner, Hughlan W. Pope, and David Brotherton pp 387 - 388; DOI: 10.1021/jm00327a024 |
2-Methacryloxytropones. Intermediates for the Synthesis of Biologically Active Polymers Robert J. Cornell and L. Guy Donaruma pp 388 - 390; DOI: 10.1021/jm00327a025 |
Improved Synthesis of Oxotremorine John L. Archibald pp 390 - 390; DOI: 10.1021/jm00327a026 |
Benzylidene Derivatives of Indene and Cyclopentadiene Carl Tabb Bahner, Harold Kinder, David Brotherton, John Spiggle, and Lee Gutman pp 390 - 392; DOI: 10.1021/jm00327a027 |
Nuclear Magnetic Resonance Spectra of Phenothiazines. Chemical Shift Data J. Cymerman Craig, D. E. Green, S. K. Roy, L. H. Piette, and Kay O. Loeffler pp 392 - 395; DOI: 10.1021/jm00327a028 |
The Synthesis, Proof of Structure, and Biological Activity of Some Monosubstituted Aminoguanidines J. Augstein, S. M. Green, A. R. Katritzky, and A. M. Monro pp 395 - 397; DOI: 10.1021/jm00327a029 |
Styrylquinoline Analogs from Heterocyclic Carboxaldehydes Carl Tabb Bahner, Harold Kinder, and Lee Gutman pp 397 - 398; DOI: 10.1021/jm00327a030 |
α- and γ-Glutamyl Derivatives of Aminobenzoic Acids Rodney F. Lloyd, Charles G. Skinner, William Shive, and R. John Stedman pp 398 - 400; DOI: 10.1021/jm00327a031 |
Synthesis of N,N-Bis(2-haloethyl) Aliphatic Amides Carlos H. Gaozza pp 400 - 401; DOI: 10.1021/jm00327a032 |
Agents Affecting Lipid Metabolism. XVI. The Synthesis of Analogs of trans-1,4-Bis(2-chlorobenzylaminomethyl)cyclohexane Leslie G. Humber pp 401 - 404; DOI: 10.1021/jm00327a033 |
A Convenient Synthesis of 5-Hydroxy-2-methyltryptophan Frederick Leonard and Walter Tschannen pp 404 - 405; DOI: 10.1021/jm00327a034 |
The Synthesis of Disalicyl Alcohols Jose Philip and John A. McLean pp 405 - 405; DOI: 10.1021/jm00327a035 |
Aromatic Fluorine Compounds. XIII. Substituted N-Phenylglycine Ethyl Esters and Hydrazides G. C. Finger, D. R. Dickerson, L. D. Starr, and D. E. Orlopp pp 405 - 407; DOI: 10.1021/jm00327a036 |
Green Medicine. The Search for Plants that Heal. Alfred Burger pp 407 - 408; DOI: 10.1021/jm00327a037 |
Infrared Absorption Spectroscopy. A. R. Patel pp 408 - 408; DOI: 10.1021/jm00327a038 |
Application of NMR Spectroscopy in Organic Chemistry. Robert A. Pages pp 408 - 408; DOI: 10.1021/jm00327a039 |
Medical Pharmacology. Daniel T. Watts pp 408 - 408; DOI: 10.1021/jm00327a040 |
The Preparation and Pharmacology of Some 3-Desoxyestratrienes. Lipid-Shifting and Estrogenic Effects Arthur H. Goldkamp, Willard M. Hoehn, Richard A. Mikulec, Ehard F. Nutting, and Donald L. Cook pp 409 - 414; DOI: 10.1021/jm00328a001 |
Synthetic Antigonadotropins. IV. Bromotriphenylethylenes H. H. Fox, J. T. Gibas, H. L. Lee, and A. Boris pp 415 - 416; DOI: 10.1021/jm00328a002 |
Action of Some Steroids on the Central Nervous System of the Mouse. I. Synthetic Methods J. D. Cocker, J. Elks, P. J. May, F. A. Nice, G. H. Phillipps, and W. F. Wall pp 417 - 425; DOI: 10.1021/jm00328a003 |
Action of Some Steroids on the Central Nervous System of the Mouse. II. Pharmacology R. M. Atkinson, B. Davis, M. A. Pratt, Helen M. Sharpe, and E. G. Tomich pp 426 - 432; DOI: 10.1021/jm00328a004 |
Synthesis of cis- and trans-2-Phenoxycyclopropylamines and Related Compounds Jacob Finkelstein, Elliot Chiang, and John Lee pp 432 - 439; DOI: 10.1021/jm00328a005 |
Amine Oxidases. XXI. A Rapid Method for the Determination of the Activity of Monoamine Oxidase and Monoamine Oxidase Inhibitors Verena Zeller, Gollamudi Ramachander, and E. Albert Zeller pp 440 - 443; DOI: 10.1021/jm00328a006 |
Synthesis of Compounds with Potential Psychotomimetic Activity. III1,2a Robert J. Adamski and Joseph G. Cannon pp 444 - 446; DOI: 10.1021/jm00328a007 |
Hydroxylamine Chemistry. V. Aralkoxyguanidines D. G. Martin, E. L. Schumann, W. Weldkamp, and H. Keasling pp 446 - 456; DOI: 10.1021/jm00328a008 |
Hydroxylamine Chemistry. V. Aralkoxyguanidines D. G. Martin, E. L. Schumann, W. Veldkamp, and H. Keasling pp 456 - 459; DOI: 10.1021/jm00328a009 |
Synthesis and Preliminary Pharmacology of Some 1-Methylindoles Robert G. Taborsky, Peter Delvigs, Irvine H. Page, and Neville Crawford pp 460 - 466; DOI: 10.1021/jm00328a010 |
Stereochemistry of d-3,4-Dimethyl-2-phenylmorpholine (Phendimetrazine) D. Dvornik and G. Schilling pp 466 - 469; DOI: 10.1021/jm00328a011 |
The Synthesis of Thyromimetic Substances and Potential Inhibitors of Thyroxine Charles M. Buess, Tullio Giudici, Norman Kharasch, William King, D. David Lawson, and N. N. Saha pp 469 - 474; DOI: 10.1021/jm00328a012 |
Hypocholesterolemic Agents. Thyroalkanols W. J. Wechter, W. A. Phillips, and F. Kagan pp 474 - 478; DOI: 10.1021/jm00328a013 |
The Synthesis of Tenuazonic and Congeneric Tetramic Acids Stanton A. Harris, Linda V. Fisher, and Karl Folkers pp 478 - 482; DOI: 10.1021/jm00328a014 |
Antitumor, Cytotoxic, and Antibacterial Activities of Tenuazonic Acid and Congeneric Tetramic Acids C. O. Gitterman pp 483 - 486; DOI: 10.1021/jm00328a015 |
Polynucleotides. III.1 Synthesis of (3′→5′)-Linked Diribonucleoside Phosphates Containing 3- and 5-Methyluracil Roosevelt Thedford, Maurice H. Fleysher, and Ross H. Hall pp 486 - 491; DOI: 10.1021/jm00328a016 |
Derivatives of Fluorene. XXI. New Halogenofluorenes. II.1a Further Potential Antitumor Agents Hsi-Lung Pan and T. Lloyd Fletcher pp 491 - 497; DOI: 10.1021/jm00328a017 |
Hexahydropyrimidines. V.1 A Study of 2-Substituted 1,3-Bis(α-cyanobenzyl)-hexahydropyrimidines and 2-Substituted 1,3-Bis(α-cyano-p-methoxybenzyl)-hexahydropyrimidines as Prospective Antitumor Agents2 John H. Billman and M. Sami Khan pp 498 - 499; DOI: 10.1021/jm00328a018 |
Synthesis of Methyl DL-3-Phthalimido-5-oxo-6-diazohexanoate Loren L. Braun and Roger M. Layton pp 500 - 502; DOI: 10.1021/jm00328a019 |
Enzyme Inhibitors. VIII. Studies on the Mode of Binding of Some 6-Substituted 9-(Hydroxyalkyl)purines to Adenosine Deaminase Howard J. Schaeffer, David Vogel, and Robert Vince pp 502 - 506; DOI: 10.1021/jm00328a020 |
Enzyme Inhibitors. IX. Hydrophobic Interactions of Some 9-Alkyladenines with Adenosine Deaminase Howard J. Schaeffer and David Vogel pp 507 - 509; DOI: 10.1021/jm00328a021 |
Glutamic Acid Analogs. The Synthesis of 3-Alkylgutamic Acids and 4-Alkylpyroglutamic Acids Yoon C. Kim and George H. Cocolas pp 509 - 513; DOI: 10.1021/jm00328a022 |
The Metabolite of 3′,5′-Dichloro-4-amino-4-deoxy-N10-methylpteroylglutamic Acid (Dichloromethotrexate) Ti Li Loo and Richard H. Adamson pp 513 - 515; DOI: 10.1021/jm00328a023 |
Synthesis and Pharmacological Action of 3-Amino-2,1-benzisothiazoles Robert F. Meyer, Betty L. Cummings, Paul Bass, and H. O. J. Collier pp 515 - 519; DOI: 10.1021/jm00328a024 |
The Metabolism of N-Alkyl-4-bromobenzenesulfonamides in the Mouse. Correlation with Anticonvulsant Activity David L. Smith, Hugh H. Keasling, and Arlington A. Forist pp 520 - 524; DOI: 10.1021/jm00328a025 |
exo-3-Chloro-endo-6-cyano-2-norbornanone O-(Methylcarbamoyl)oxime. A New Type of Methylcarbamate with Acaricidal Activity Linwood K. Payne, Harry A. Stansbury, and Mathias H. J. Weiden pp 525 - 528; DOI: 10.1021/jm00328a026 |
Chemical Structure and Pharmacological Activity of Glycine Derivatives. Influence of Disubstitution of the Amine Function of Glycine Esters and Hydrazides Richard Rips, Christian Derappe, and Pierre Magnin pp 529 - 531; DOI: 10.1021/jm00328a027 |
3-Piperonylsydnone. A New Type of Antimalarial Agent Wayne H. Nyberg and C. C. Cheng pp 531 - 533; DOI: 10.1021/jm00328a028 |
Thyroxine Analogs. XV.1 Synthesis and Antigoitrogenic Activity of the 3′-t-Butyl Analog of 3,5,3′-Triiodo-L-thyronine and Its O-Methyl Ether Eugene C. Jorgensen and James A. W. Reid pp 533 - 536; DOI: 10.1021/jm00328a029 |
17-Chloroethynylated Steroids. III. The Synthesis of 17α-Chloroethynyl-5,7,9-estratrien-17β-ol-3-one John Hannah and John H. Fried pp 536 - 537; DOI: 10.1021/jm00328a030 |
A-Nor Oxa Steroids Seymour D. Levine pp 537 - 539; DOI: 10.1021/jm00328a031 |
Synthesis of Potential Antidiabetic Agents. 1-p-Tolylsulfonyl-2-benzimidazolinones and 1-p-Tolylsulfonyl-2-benzimidazolinethiones John B. Wright pp 539 - 540; DOI: 10.1021/jm00328a032 |
Hexahydropyrimidines. VI. Some 2-{4-[N,N-Bis(2-chloroethyl)amino]aryl}- 1,3-bis(aralkyl)hexahydropyrimidines John H. Billman and John L. Meisenheimer pp 540 - 540; DOI: 10.1021/jm00328a033 |
N4-(2-Bromoethyl)-N4-ethylsulfanilamide, a Monofunctional Nitrogen Mustard with Antitumor Action P. Hebborn and D. J. Triggle pp 541 - 542; DOI: 10.1021/jm00328a034 |
Basic Ethers of Guaiacol and Thymol with a Polyoxyethylenic Chain and Their Main Pharmacological Activities. New Antitussives M. Carissimi, A. Cattaneo, R. D'Ambrosio, V. De Pascale, E. Grumelli, E. Milla, and F. Ravenna pp 542 - 545; DOI: 10.1021/jm00328a035 |
Insect Chemosterilants. II.1 N-Carbamoylaziridines Alexej B. Bořkovec and Charles W. Woods pp 545 - 547; DOI: 10.1021/jm00328a036 |
Cytotoxicity of Cardiac Principles R. B. Kelly, Edward G. Daniels, and L. Bayard Spaulding pp 547 - 548; DOI: 10.1021/jm00328a037 |
The Relationship between Structure and Anticonvulsant Activity in a Series of Benzenesulfonamides H. H. Keasling, E. L. Schumann, and W. Veldkamp pp 548 - 550; DOI: 10.1021/jm00328a038 |
Some 2,3,6-Trisubstituted Quinazolones K. Kishor, R. C. Arora, and Surendra S. Parmar pp 550 - 551; DOI: 10.1021/jm00328a039 |
Derivatives of Fluorene. XX.1a,b Fluorofluorenes. V. New Difluoro-2-acetamidofluorenes for the Study of Carcinogenic Mechanisms Moses J. Namkung, T. Lloyd Fletcher, and William H. Wetzel pp 551 - 554; DOI: 10.1021/jm00328a040 |
The Synthesis of DL-p-(Hydroxymethyl)phenylalanine G. W. E. Plaut pp 554 - 555; DOI: 10.1021/jm00328a041 |
Coupling Reactions in the Synthesis of Amitriptyline R. D. Hoffsommer, D. Taub, and N. L. Wendler pp 555 - 556; DOI: 10.1021/jm00328a042 |
Psychopharmacological Agents. Volume I. Alfred Burger pp 556 - 556; DOI: 10.1021/jm00328a043 |
N-Allylnorapomorphine Jerome F. Hensiak, Joseph G. Cannon, and Allan M. Burkman pp 557 - 559; DOI: 10.1021/jm00329a001 |
Constitution and Analgetic Activity of a New Product in the Benzomorphan Synthesis Bhuwan C. Joshi, Everette L. May, H. M. Fales, J. W. Daly, and A. E. Jacobson pp 559 - 563; DOI: 10.1021/jm00329a002 |
Structures Related to Morphine. XXXI.1 2′-Substituted Benzomorphans Arthur E. Jacobson and Everette L. May pp 563 - 566; DOI: 10.1021/jm00329a003 |
Analgesics. Some Substituted 2,3-Dihydro-4-quinolones M. S. Atwal, L. Bauer, S. N. Dixit, J. E. Gearien, and R. W. Morris pp 566 - 571; DOI: 10.1021/jm00329a004 |
Chemistry and Pharmacology of Some Esters Derived from Basic Alcohols F. P. Doyle, M. D. Mehta, R. Ward, J. Bainbridge, and D. M. Brown pp 571 - 576; DOI: 10.1021/jm00329a005 |
Cardiac Glycosides and Aglycones by Synthesis and Microbiological Conversion Francis G. Henderson and K. K. Chen pp 577 - 579; DOI: 10.1021/jm00329a006 |
The Adamantyl Group in Medicinal Agents. II. Anabolic Steroid 17β-Adamantoates Richard T. Rapala, Russell J. Kraay, and Koert Gerzon pp 580 - 583; DOI: 10.1021/jm00329a007 |
Synthesis of α-(p-Aminophenyl)- and α-(p-Chlorophenyl)-β-arylpropionitriles by Catalytic Reduction of Stilbenenitriles Gordon N. Walker pp 583 - 588; DOI: 10.1021/jm00329a008 |
Synthesis and Pharmacological Evaluation of α,α-Disubstituted Derivatives of Phenylacetonitrile and 1-Naphthylacetonitrile Silvano Casadio, Gianfranco Pala, Elda Crescenzi, Tiberio Bruzzese, Ernesta Marazzi-Uberti, and Germano Coppi pp 589 - 593; DOI: 10.1021/jm00329a009 |
Synthesis and Pharmacological Evaluation of α,α-Disubstituted Derivatives of Phenylacetamide and 1-Naphthylacetamide Silvano Casadio, Gianfranco Pala, Tiberio Bruzzese, Elda Crescenzi, Ernesta Marazzi-Uberti, and Germano Coppi pp 594 - 598; DOI: 10.1021/jm00329a010 |
Nonsteroidal Antiinflammatory Agents. Some Arylacetic Acids G. J. Durant, G. M. Smith, R. G. W. Spickett, and E. Szarvasi pp 598 - 603; DOI: 10.1021/jm00329a011 |
Silicon-Substituted Medicinal Agents. Silacarbamates Related to Meprobamate Ralph J. Fessenden and Marvin D. Coon pp 604 - 608; DOI: 10.1021/jm00329a012 |
A New Concept on the Mode of Interaction of Narcotic Analgesics with Receptors Philip S. Portoghese pp 609 - 616; DOI: 10.1021/jm00329a013 |
Stereochemical Factors Related to the Potency of Anticholinergic Psychotomimetic Drugs Norman W. Gabel and Leo G. Abood pp 616 - 619; DOI: 10.1021/jm00329a014 |
Compounds Affecting the Central Nervous System. I. 4-Piperidones and Related Compounds C. R. Ganellin and R. G. W. Spickett pp 619 - 625; DOI: 10.1021/jm00329a015 |
Synthesis of New 3-(Pyridylmethylene)-, 3-(Pyridylmethyl)-, 3-(Piperidylmethyl)-, and 3-(β-Alkylaminoethyl)-2-indolinones. The Reduction of Isoindogenides, Nitro Compounds, and Pyridines in a Series of 2-Indolinones Gordon N. Walker, Ronald T. Smith, and Barbara N. Weaver pp 626 - 637; DOI: 10.1021/jm00329a016 |
Pyrazine Diuretics. I. N-Amidino-3-amino-6-halopyrazinecarboxamides John B. Bicking, James W. Mason, Otto W. Woltersdorf, James H. Jones, Sara F. Kwong, Charles M. Robb, and Edward J. Cragoe pp 638 - 642; DOI: 10.1021/jm00329a017 |
Physiologically Active Compounds. VI. Cyclic Amino Thiolesters of Substituted Chloroacetic, Benzilic, and Glycolic Acids Calvin A. Buehler, Shelby F. Thames, L. G. Abood, and J. H. Biel pp 643 - 647; DOI: 10.1021/jm00329a018 |
Effect of Organic Compounds on Reproductive Processes. I. Alkylating Agents from Octamethylenediamine and Various Xylylenediamines W. A. Skinner, H. C. Tong, T. E. Shellenberger, and G. W. Newell pp 647 - 650; DOI: 10.1021/jm00329a019 |
Some Amino and Ammonio Nitrogen Mustard Analogs Charles C. Price, Guglielmo Kabas, and Isao Nakata pp 650 - 655; DOI: 10.1021/jm00329a020 |
Diazo, Bromo, and Mesyloxy Ketones as Biological Alkylating Agents T. Nogrady, T. W. Doyle, and L. Morris pp 656 - 659; DOI: 10.1021/jm00329a021 |
3′-Deoxynucleosides. II. Purine 3′-Deoxynucleosides Edward Walton, Frederick W. Holly, George E. Boxer, Ruth F. Nutt, and Susan R. Jenkins pp 659 - 663; DOI: 10.1021/jm00329a022 |
Relation of Structure to Activity of Purine 3′-Deoxynucleosides in KB Cell and Chick Embryo Fibroblast Cell Cultures C. O. Gitterman, R. W. Burg, G. E. Boxer, D. Meltz, and J. Hitt pp 664 - 667; DOI: 10.1021/jm00329a023 |
The Synthesis and Properties of 6-Mercaptomethylpurine and Derivatives Alfredo Giner-Sorolla and Aaron Bendich pp 667 - 672; DOI: 10.1021/jm00329a024 |
Structural Studies of an Active Principle from Croton tiglium L. Eugene R. Arroyo and J. Holcomb pp 672 - 675; DOI: 10.1021/jm00329a025 |
Antiviral Chemotherapy. I. The Activity of Pyridine and Quinoline Derivatives against Neurovaccinia in Mice D. H. Jones, R. Slack, S. Squires, and K. R. H. Wooldridge pp 676 - 680; DOI: 10.1021/jm00329a026 |
Antiviral Chemotherapy. II. Structure-Activity Relationships in a Series of Isothiazolealdehyde and Ketone Thiosemicarbazones M. P. L. Caton, D. H. Jones, R. Slack, S. Squires, and K. R. H. Wooldridge pp 680 - 683; DOI: 10.1021/jm00329a027 |
Aminooxy Derivatives. IV. Antimicrobial Activity of Some O-Ethers of 4,6-Diamino-1,2-dihydro-1-hydroxy-2-substituted 1,3,5-Triazines P. Mamalis, L. Jeffries, S. A. Price, M. J. Rix, and D. J. Outred pp 684 - 691; DOI: 10.1021/jm00329a028 |
New Sulfonamides J. M. Loynes, H. F. Ridley, and R. G. W. Spickett pp 691 - 694; DOI: 10.1021/jm00329a029 |
Structures Related to Morphine. XXX.1 N-Hexyl- and 5-Butyl-, -Amyl-, and -Hexyl-6,7-benzomorphans Bhuwan C. Joshi, Colin F. Chignell, and Everette L. May pp 694 - 696; DOI: 10.1021/jm00329a030 |
Structures Related to Morphine. XXXII.1 α- and β-2,9-Dimethyl-5-propyl-6,7-benzomorphan from 3-Methyl-4-propylpyridine Bhuwan C. Joshi and Everette L. May pp 696 - 697; DOI: 10.1021/jm00329a031 |
1-(3-Phenylpropyl)-2-methyl-6,7-methylenedioxy-8-methoxy-1,2,3,4- tetrahydroisoquinoline, a Pharmacologically Active Narcotine Derivative Arthur E. Jacobson pp 697 - 698; DOI: 10.1021/jm00329a032 |
Structure-Activity Relationships in Antiinflammatory and Analgesic Compounds Chemically Related to α-Isopropyl-α-(2-dimethylaminoethyl)-1-naphthylacetamide G. Pala, S. Casadio, T. Bruzzese, E. Crescenzi, and E. Marazzi-Uberti pp 698 - 700; DOI: 10.1021/jm00329a033 |
9-(2-Aminoethyl)-2,3-dihydro-1H-pyrrolo[1,2-a]-indoles, New Tryptamine Analogs William A. Remers and Martin J. Weiss pp 700 - 702; DOI: 10.1021/jm00329a034 |
Isomeric Benzyldiaminodihydrotriazines Howard Newman and Edward L. Moon pp 702 - 704; DOI: 10.1021/jm00329a035 |
Spiranes. IX. Amides of 3,9-Dicarboxy-2,4,8,10-tetraoxaspiro[5.5]undecane Leonard M. Rice and Charles H. Grogan pp 704 - 705; DOI: 10.1021/jm00329a036 |
The Structure-Activity Relationship in Penicillins Corwin Hansch and Edna W. Deutsch pp 705 - 706; DOI: 10.1021/jm00329a037 |
Dihydrazides, a New Class of Anthelmintics Raymond Cavier and Richard Rips pp 706 - 708; DOI: 10.1021/jm00329a038 |
Deaza Analogs of 6-Mercaptopurine John A. Montgomery and Kathleen Hewson pp 708 - 710; DOI: 10.1021/jm00329a039 |
Enzyme Inhibitors. X. A Reinvestigation of the Alkylation of 6-Chloropurine by 3-Bromo-1-propanol Howard J. Schaeffer and Robert Vince pp 710 - 712; DOI: 10.1021/jm00329a040 |
3′-Iodo-4-amino-4-deoxypteroylglutamic Acid (3′-Iodoaminopterin) Ti Li Loo, Robert L. Dion, Richard H. Adamson, Michael A. Chirigos, and Roy L. Kisliuk pp 713 - 715; DOI: 10.1021/jm00329a041 |
Bis(2-chloroalkyl)amides of Acylated Amino Acids. Modified Nitrogen Mustards Irving Levi, Harold Blondal, J. William R. Weed, Alan C. Frosst, H. Christine Reilly, Franz A. Schmid, Kanematsu Sugiura, George S. Tarnowski, and C. Chester Stock pp 715 - 718; DOI: 10.1021/jm00329a042 |
Chloroalkyl-N-sulfinylamines Walter T. Smith, Wen-Yean Chen, and Myron Linfield pp 718 - 719; DOI: 10.1021/jm00329a043 |
Anticholinergic Agents. Esters of 4-Dialkyl- (or 4-Polymethylene-) amino-2-butynols Robert F. Majewski, Kenneth N. Campbell, Stanley Dykstra, Robert Covington, and Jack C. Simms pp 719 - 720; DOI: 10.1021/jm00329a044 |
New Antifertility Agents. 2,3-Diphenylbenzofurans P. K. Grover, H. P. S. Chawla, Nitya Anand, V. P. Kamboj, and Amiya B. Kar pp 720 - 721; DOI: 10.1021/jm00329a045 |
5-Aryl-1,3-dihydro-2H-pyrido-1,4-diazepin-2-ones Ruddy Littell and Duff S. Allen pp 722 - 724; DOI: 10.1021/jm00329a046 |
Mammalian Antifertility Agents. II. Basic Ethers of 3,4-Diphenylcoumarins Daniel Lednicer, Stanley C. Lyster, and Gordon W. Duncan pp 725 - 726; DOI: 10.1021/jm00329a047 |
3′-Fluorofolic Acid John A. Montgomery, Kathleen Hewson, and J. Robert Piper pp 727 - 728; DOI: 10.1021/jm00329a048 |
The Synthesis of Some Benzimidazole and Oxygen Analogs of Ethyl Pteroylglutamate Bruce I. Dittmar and Allan R. Day pp 728 - 728; DOI: 10.1021/jm00329a049 |
Myelographic Agents. I. Iodobenzoates J. E. Siggins, J. H. Ackerman, and A. A. Larsen pp 728 - 730; DOI: 10.1021/jm00329a050 |
The Synthesis of Ethyl p-Nitrophenyl α-Acetoxyalkylphosphonates L. S. Hafner, J. E. Brown, M. V. Garrison, and B. H. Alexander pp 730 - 731; DOI: 10.1021/jm00329a051 |
3-Phenylphthalimidines Price Truitt, Linda Reeves Brammer, and Linda Truitt Creagh pp 731 - 732; DOI: 10.1021/jm00329a052 |
Some Compounds Derived from 1-Cyano- and 1-Bromobenzocyclobutene Joseph A. Skorcz and Frank E. Kaminski pp 732 - 734; DOI: 10.1021/jm00329a053 |
Some N-Substituted Dimethoxyphenylacetamides and Dimethoxyphenylethylamines C. G. Stuckwisch and Janice S. Hilliard pp 734 - 735; DOI: 10.1021/jm00329a054 |
Drugs of Choice 1964-1965. John A. Owen pp 735 - 735; DOI: 10.1021/jm00329a055 |
The National Formulary, Twelfth Edition. Warren E. Weaver pp 735 - 736; DOI: 10.1021/jm00329a056 |
The Quantitative Analysis of Drugs. Anilkumar P. Parulkar pp 736 - 736; DOI: 10.1021/jm00329a057 |
Synthesis of Potential Anticancer Agents. XXXIV. Fluorobenzimidazoles and Fluorobenzotriazoles John A. Montgomery and Kathleen Hewson pp 737 - 740; DOI: 10.1021/jm00330a001 |
2-Fluoroethylamines. II.1a Biological Evaluation and Synthesis1b Abelardo P. Martinez, William W. Lee, and Leon Goodman pp 741 - 744; DOI: 10.1021/jm00330a002 |
Potential Folic Acid Antagonists. I. The Antitumor and Folic Acid Reductase Inhibitory Properties of 6-Substituted 2,4-Diamino-5-arylazopyrimidines J. Hampshire, P. Hebborn, A. M. Triggle, D. J. Triggle, and S. Vickers pp 745 - 749; DOI: 10.1021/jm00330a003 |
2,4-Dimethyl-5-hydroxymethylpyrimidine, a Pyridoxol Antagonist Thomas J. Schwan, Howard Tieckelmann, James F. Holland, and Bradley Bryant pp 750 - 753; DOI: 10.1021/jm00330a004 |
The Effect of Some Sulfur-Containing Pyridine Derivatives on the Carbohydrate Metabolism of Ehrlich Ascites Tumor D. R. Grassetti, M. E. Brokke, and J. F. Murray pp 753 - 756; DOI: 10.1021/jm00330a005 |
A Highly Reactive Sulfur Mustard Gas Derivative for Localized Infusion Studies W. Davis and W. C. J. Ross pp 757 - 759; DOI: 10.1021/jm00330a006 |
Reactivity of Some 2-p-Nitrophenoxy-1,3,2-dioxaphospholane 2-Oxides and -dioxaphosphorinane 2-Oxides T. R. Fukuto and R. L. Metcalf pp 759 - 762; DOI: 10.1021/jm00330a007 |
Potential Antiradiation Drugs. II.1 2-Amino-1-alkanethiols, 1-Amino-2-alkanethiols, 2-Thiazolines, and 2-Thiazoline-2-thiols2 G. Richard Handrick, Edward R. Atkinson, Felix E. Granchelli, and Robert J. Bruni pp 762 - 766; DOI: 10.1021/jm00330a008 |
Sulfamylurea Hypoglycemic Agents. I. Synthesis and Screening J. M. McManus, J. W. McFarland, C. F. Gerber, W. M. McLamore, and G. D. Laubach pp 766 - 776; DOI: 10.1021/jm00330a009 |
Sulfamylurea Hypoglycemic Agents. II. Drug Dynamic Studies Edward H. Wiseman, J. N. Pereira, K. F. Finger, and Rex Pinson pp 777 - 781; DOI: 10.1021/jm00330a010 |
Sulfamylurea Hypoglycemic Agents. III. Tetrasubstituted Sulfamylureas and N-Sulfamylcarbamates J. W. McFarland, C. F. Gerber, and W. M. McLamore pp 781 - 784; DOI: 10.1021/jm00330a011 |
Sulfanilamido-s-triazines. I. Synthesis of 2-Sulfanilamido-4,6-diethyl-s-triazine and Related Compounds W. E. Taft, H. M. Krazinski, F. C. Schaefer, and R. G. Shepherd pp 784 - 789; DOI: 10.1021/jm00330a012 |
Rifamycins. XLI.1 A New Class of Active Semisynthetic Rifamycins. N-Substituted Aminomethyl Derivatives of Rifamycin SV2 N. Maggi, V. Arioli, and P. Sensi pp 790 - 793; DOI: 10.1021/jm00330a013 |
Derivatives of 6-Aminopenicillanic Acid. VI. Synthesis of Some Derivatives of 6-Aminothiopenicillanic Acid W. J. Gottstein, R. B. Babel, L. B. Crast, J. M. Essery, R. R. Fraser, J. C. Godfrey, C. T. Holdrege, W. F. Minor, M. E. Neubert, C. A. Panetta, and L. C. Cheney pp 794 - 797; DOI: 10.1021/jm00330a014 |
Studies on 2-(α-Hydroxybenzyl)benzimidazole (HBB) Analogs. I. Synthesis of 8-(α-Hydroxybenzyl)purines, the Diaza Analogs of HBB William J. Haggerty, Robert H. Springer, and C. C. Cheng pp 797 - 802; DOI: 10.1021/jm00330a015 |
Substituted 5,6-Dihydro-2-(2-, 3-, and 4-pyridyl)-4H-1,3,4-oxadiazines Donald L. Trepanier, Paul E. Krieger, and John N. Eble pp 802 - 807; DOI: 10.1021/jm00330a016 |
New Sedative and Hypotensive 3-Substituted 2,4(1H,3H)-Quinazolinediones Shin Hayao, Herbert J. Havera, Wallace G. Strycker, T. J. Leipzig, Richard A. Kulp, and Harold E. Hartzler pp 807 - 811; DOI: 10.1021/jm00330a017 |
Unnatural Amino Acids. I. 3-Carboxytyrosine Derivatives Frederick Leonard, Abraham Wajngurt, Walter Tschannen, and Fred B. Block pp 812 - 815; DOI: 10.1021/jm00330a018 |
Quinazolines and 1,4-Benzodiazepines. XXV.1 Structure-Activity Relationships of Aminoalkyl-Substituted 1,4-Benzodiazepin-2-ones L. H. Sternbach, G. A. Archer, J. V. Earley, R. Ian Fryer, E. Reeder, N. Wasyliw, L. O. Randall, and R Banzger pp 815 - 821; DOI: 10.1021/jm00330a019 |
Further Syntheses in the Study of Structure-Activity Relationships of Neuropharmacologically Active Amino Acids K. S. Cheah and J. C. Watkins pp 821 - 824; DOI: 10.1021/jm00330a020 |
Spiranes. X. Aminospiranes1,2a Leonard M. Rice, Edward C. Dobbs, and Charles H. Grogan pp 825 - 829; DOI: 10.1021/jm00330a021 |
Structure-Activity Relationships in the Cyproheptadine Series Edward L. Engelhardt, Howard C. Zell, Walfred S. Saari, Marcia E. Christy, C. Dylion Colton, Clement A. Stone, John M. Stavorski, Herbert C. Wenger, and Carl T. Ludden pp 829 - 835; DOI: 10.1021/jm00330a022 |
Compounds Affecting the Central Nervous System. III. Substituted 1,1-Diaryl-t-aminopropanols and Related Compounds D. I. Barron, G. H. Hall, I. L. Natoff, H. F. Ridley, R. G. W. Spickett, and D. K. Vallance pp 836 - 841; DOI: 10.1021/jm00330a023 |
Synthesis and Cholinergic Effects of Certain N-Methoxylated Quaternary Compounds Laszlo L. Darko, Joseph G. Cannon, John P. Long, and Thomas F. Burks pp 841 - 844; DOI: 10.1021/jm00330a024 |
Analogs of Parasympathetic Neuroeffectors. III. Synthesis and Study of Cholineselenol and Related Compounds Wolfgang H. H. Günther and Henry G. Mautner pp 845 - 847; DOI: 10.1021/jm00330a025 |
Structure-Activity Relationship of Some New Analogs of Pethidine D. G. Hardy, R. E. Lister, and E. S. Stern pp 847 - 851; DOI: 10.1021/jm00330a026 |
4-Substituted Piperidines. II. Reaction of 1-Benzyl-4-cyano-4-t-aminopiperidines with Organometallic Compounds Bert Hermans, Paul Van Daele, Cornelis Van De Westeringh, Cyriel Van Der Eycken, Jozef Boey, and Paul A. J. Janssen pp 851 - 855; DOI: 10.1021/jm00330a027 |
6-Hydroxyindoles and the Metabolism of Melatonin Robert G. Taborsky, Peter Delvigs, and Irvine H. Page pp 855 - 858; DOI: 10.1021/jm00330a028 |
In Vitro Inhibition Studies with Homogeneous Monoamine Oxidases Alfred Burger and Sakari Nara pp 859 - 862; DOI: 10.1021/jm00330a029 |
Potential Antiradiation Agents.1a Preparation and Polymerization of Monomeric Thiazolidines1b,c C. G. Overberger, H. Ringsdorf, and B. Avchen pp 862 - 864; DOI: 10.1021/jm00330a030 |
Substituted 2-Aminothiosulfuric Acids Derived from α-Amino Acids Herman Gershon and Raymond Rodin pp 864 - 866; DOI: 10.1021/jm00330a031 |
2-Trifluoromethyladenosine G. Gough and M. H. Maguire pp 866 - 867; DOI: 10.1021/jm00330a032 |
Antituberculous Compounds. XXII.1 Monoalkylaminobenzothioamides Shichiro Kakimoto and Ikuko Tone pp 867 - 868; DOI: 10.1021/jm00330a033 |
Antituberculous Compounds. XXIII.1 Alkyl- and Acylisonicotinic Acid Hydrazides Shichiro Kakimoto and Ikuko Tone pp 868 - 868; DOI: 10.1021/jm00330a034 |
The Use of Substituent Constants in the Correlation of Demethylation Rates Corwin Hansch, A. Ruth Steward, and Junkichi Iwasa pp 868 - 870; DOI: 10.1021/jm00330a035 |
Alkoxyalkyltetracyclines C. Richard Tamorria and Robert C. Esse pp 870 - 872; DOI: 10.1021/jm00330a036 |
Synthesis of Heterocyclic-Substituted Chromones and Related Compounds as Potential Anticancer Agents Dorothy Donnelly, Rosalie Geoghegan, Conor O'Brien, Eva Philbin, and T. S. Wheeler pp 872 - 875; DOI: 10.1021/jm00330a037 |
Synthetic Spasmolytic Amines George H. Cocolas, Souren Avakian, and Gustav J. Martin pp 875 - 877; DOI: 10.1021/jm00330a038 |
Amino Acid Analogs. I. Analogs of the Glutamic Acid-Proline Interconversion. III. Substituted 2-Acetamido-4-benzoylbutyric Acids and 5-Phenylprolines Herman Gershon, Alfred Scala, and Raulo Parmegiani pp 877 - 881; DOI: 10.1021/jm00330a039 |
Reduction of Steroidal Enamines with Potassium Borohydride Arvin P. Shroff pp 881 - 883; DOI: 10.1021/jm00330a040 |
Some 3,4,5-Trimethoxyphenyl Analogs of Anticonvulsants Vasant S. Palkar and Pierre F. Smith pp 883 - 884; DOI: 10.1021/jm00330a041 |
Synthesis of Some Hydroxylamine Derivatives of Pyrimidines and Purines Pauline K. Chang pp 884 - 884; DOI: 10.1021/jm00330a042 |
Quinoxaline Sulfonamides S. H. Dandegaonker and C. K. Mesta pp 884 - 886; DOI: 10.1021/jm00330a043 |
Transformation Products of 5H-Dibenzo-[αd]-10,11-dihydrocyclohepten-5-one H. L. Slates and N. L. Wendler pp 886 - 886; DOI: 10.1021/jm00330a044 |
The Synthesis of Aryloxyureas Victor J. Bauer and Harry P. Dalalian pp 886 - 887; DOI: 10.1021/jm00330a045 |
1-Acyl-1-alkoxy-3-(p-tolylsulfonyl)ureas James H. Cooley and J. Dana McCown pp 887 - 888; DOI: 10.1021/jm00330a046 |
Monothiophenyl Malonate John C. Howard, Michael C. Lin, Patricia Matthews, and Sam A. Singal pp 888 - 888; DOI: 10.1021/jm00330a047 |
The Reaction of Chloramine with Mercaptopyridine and Mercaptopyrimidine Derivatives Thomas J. Hurley and Martin A. Robinson pp 888 - 889; DOI: 10.1021/jm00330a048 |
Potential Inhibitors of Cancerous Growth. V. Substituted Benzylidene Derivatives of D-Ribose as Synthetic Intermediates W. J. Serfontein, G. J. Lourens, and H. L. De Waal pp 889 - 891; DOI: 10.1021/jm00330a049 |
Some New Arylphosphonic and Diarylphosphinic Acids Leon D. Freedman and G. O. Doak pp 891 - 892; DOI: 10.1021/jm00330a050 |
Substituted 1,4-Diazepin-2-ones Ruddy Littell and Duff S. Allen pp 892 - 893; DOI: 10.1021/jm00330a051 |
Book Review - Screening Methods in Pharmacology. Alfred Burger pp 894 - 894; DOI: 10.1021/jm00330a052 |
Addtions and Corrections - Some 2-Substituted Aminopurines and Purine Analogs. R. M. Cresswell, T. Strauss, and George Bosworth Brown pp 894 - 895; DOI: 10.1021/jm00330a053 |
Additions and Corrections - Derivatives of Fluorenes. XVIII. New Halogenofluorenes. I. Potential Antitumor Agents. Hsi-Lung Pan, and T. Lloyd Fletcher pp 894 - 894; DOI: 10.1021/jm00330a600 |
Additions and Corrections - 4-Substituted Piperidines. I. Derivativesof 4-t-Aminopiperidinecarboxamines. C. van de Westeringh, P. Van Daele, B. Hermans, C. Van der Eycken, J. Boey, and P. A. J. Janssen pp 894 - 894; DOI: 10.1021/jm00330a601 |
Additions and Corrections - Structure Studies on Vancomycin. Frederick J. Marshall pp 894 - 894; DOI: 10.1021/jm00330a602 |
Additions and Corrections - Synthesis and Biological Evaluation of Water-Soluble 2-Boronoethylthio Compounds. D. S. Matteson, A. H. Soloway, D. W. Tomlinson, J. D. Campbell, and G. A. Nixon pp 894 - 894; DOI: 10.1021/jm00330a603 |
Additions and Corrections - 17α-Methandrostane-3α,17β-diol K. R. Bharucha, and F. M. Martin pp 895 - 895; DOI: 10.1021/jm00330a604 |
Additions and Corrections - Hydroxy-, Nitro-, Amino-, and Methoxy-4-(4-dimethylaminostyryl)-quinolines. C. T. Bahner, D. Brotherton, W. H. Chapman, Jr., W. Longmire, H. B. Orr, L. M. Rives, E. B. Senter, and W. Yee pp 895 - 895; DOI: 10.1021/jm00330a605 |
Additions and Corrections - Review of "Advances in Drug Research" Alfred Burger pp 895 - 895; DOI: 10.1021/jm00330a606 |
Additions and Corrections - Phosphorylated Benzenesulfonamides as Animal Systemic Insecticides F. A. Wagner, Jr., R. W. Baer, and G. Berkelhammer pp 895 - 895; DOI: 10.1021/jm00330a607 |
Additions and Corrections - Adrenergic Blocking Agents Derived from 1,4-Benzodiozan. J. Augstein, S. M. Green, A. M. Munro, G. W. H. Potter, C. R. Worthing, and T. L. Wrigley pp 895 - 895; DOI: 10.1021/jm00330a608 |